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Formula
C22H24ClN5O2
MW
425.92
Purity
>97%
Solubility (DMSO Mg/MI)
40
Bio Chemical Notes
Dopamine D2 antagonist with Ki = 6.7 microM. An antidopaminergic drug which is used to supress nausea and vomiting, it has been shown to be effective as a prokinetic agent for promoting lactation. Ref: J Neurochem 1988; 51 (5); 1510-1515.
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