Product Details
Formula
C16H14ClN3O2
MW
315.76
Purity
>97%
Solubility (DMSO Mg/MI)
20
Storage (Powder)
3 Years -20°C
Storage (Solvent)
1 Year -80°C
Indication
Glioblastomas and in Breast, Lung and Ovarian Cancers
Mode Of Action
inhibitor
Target Name
Epidermal growth factor receptor (EGFR)
Research Area
CANCER
Research Area Sub Group
Anticancer
Pharmacology
ENZYME-LINKED RECEPTORS
Pharmacology Area Sub Group
Kinase
Bio Chemical Notes
A selective inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase, displaying IC50 = 1.26nM. Ref: JMC 2005; 48 (23); 7445-7456.
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